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Item Details
Title: ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS, VOLUME 45
By: Arun K. Ghosh (Editor), Raimund Mannhold, Hugo Kubinyi
Format: Electronic book text

List price: £168.00


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ISBN 10: 3527630953
ISBN 13: 9783527630950
Publisher: JOHN WILEY AND SONS LTD
Pub. date: 28 July, 2010
Series: Methods and Principles in Medicinal Chemistry 45
Pages: 640
Description: In this ground-breaking practical reference, the family of aspartic acid proteases is described from a drug developer's perspective. The first part provides a general introduction to the family of aspartic acid proteases, their physiological functions, molecular structure and inhibition.
Synopsis: In this ground-breaking practical reference, the family of aspartic acid proteases is described from a drug developer's perspective. The first part provides a general introduction to the family of aspartic acid proteases, their physiological functions, molecular structure and inhibition. Parts two to five present various case studies of successful protease inhibitor drug design and development, as well as current and potential uses of such inhibitors in pharmaceutical medicine, covering the major therapeutic targets HIV-1 protease, renin, beta-secretase, gamma-secretase,plasmepsins and fungal proteases. A ready reference aimed primarily at professionals in the pharmaceutical industry, as well as for anyone studying proteases and their function.
Publication: UK
Imprint: Wiley-VCH Verlag GmbH
Returns: Non-returnable
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