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Item Details
Title: TRANSPORTERS AS DRUG TARGETS
Volume: Volume 70
By: Gerhard F. Ecker (Editor), Rasmus P. Clausen (Editor), Harald H. Sitte (Editor)
Format: Hardback

List price: £131.95


We currently do not stock this item, please contact the publisher directly for further information.

ISBN 10: 3527333843
ISBN 13: 9783527333844
Publisher: WILEY-VCH VERLAG GMBH
Pub. date: 18 February, 2015
Series: Methods and Principles in Medicinal Chemistry Volume 70
Pages: 354
Description: As opposed to other books on the topic, this volume is unique in also covering emerging transporter targets. Following a general introduction to the importance of targeting transporter proteins with drugs, the book systematically presents individual transporter classes and explains their pharmacology and physiology.
Synopsis: As opposed to other books on the topic, this volume is unique in also covering emerging transporter targets. Following a general introduction to the importance of targeting transporter proteins with drugs, the book systematically presents individual transporter classes and explains their pharmacology and physiology. The text covers all transporter families with known or suspected importance as drug targets, including neurotransmitter transporters, ABC transporters, glucose transporters and organic ion transporters. The final part discusses recent advances in structural studies of transport proteins, assay methods for transport activity, and the systems biology of transporters and their regulation. With its focus on drug development issues, this authoritative overview is required reading for researchers in industry and academia targeting transport proteins for the treatment of disease.
Publication: Germany
Imprint: Blackwell Verlag GmbH
Returns: Returnable
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ANTIVIRAL DRUG STRATEGIES (HB)
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ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS (HB)
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BIO-NMR IN DRUG RESEARCH (HB)
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54
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BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54 (HB)
BIONMR IN DRUG RESEARCH, VOLUME 16
CHEMOGENOMICS IN DRUG DISCOVERY
CHEMOINFORMATICS IN DRUG DISCOVERY (HB)
CHEMOINFORMATICS IN DRUG DISCOVERY, VOLUME 23
CHEMOKINE RECEPTORS AS DRUG TARGETS (HB)
CHEMOMETRIC METHODS IN MOLECULAR DESIGN, VOLUME 2
CHIRALITY IN DRUG RESEARCH, VOLUME 33
CHIRALITY IN DRUG RESEARCH, VOLUME 33 (HB)
COMBINATORIAL CHEMISTRY
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DRUG BIOAVAILABILITY
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DRUG METABOLISM PREDICTION, VOLUME 63
DRUG METABOLISM PREDICTION, VOLUME 63
DRUG METABOLISM PREDICTION, VOLUME 63
DRUG METABOLISM PREDICTION, VOLUME 63 (HB)
DRUG SELECTIVITY
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EPIGENETIC TARGETS IN DRUG DISCOVERY
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EVOLUTIONARY ALGORITHMS IN MOLECULAR DESIGN, VOLUME 8
FRAGMENT-BASED APPROACHES IN DRUG DISCOVERY
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FRAGMENT-BASED DRUG DISCOVERY
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G PROTEIN-COUPLED RECEPTORS AS DRUG TARGETS
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HIGH-THROUGHPUT SCREENING IN DRUG DISCOVERY
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HIT AND LEAD PROFILING (HB)
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LEAD GENERATION
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LIGAND DESIGN FOR G PROTEIN-COUPLED RECEPTORS
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MASS SPECTROMETRY IN MEDICINAL CHEMISTRY
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PREDICTIVE TOXICOLOGY
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