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Item Details
Title: PHARMACOKINETICS AND METABOLISM IN DRUG DESIGN, VOLUME 51
By: Dennis A. Smith (Editor), Charlotte Allerton (Editor), Hugo Kubinyi (Editor)
Format: Hardback

List price: £116.95
Our price: £96.48
Discount:
17.5% off
You save: £20.47
ISBN 10: 3527329544
ISBN 13: 9783527329540
Availability: Usually dispatched within 1-3 weeks.
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Publisher: WILEY-VCH VERLAG GMBH
Pub. date: 4 April, 2012
Edition: 3rd Edition
Series: Methods and Principles in Medicinal Chemistry
Pages: 268
Description: A concise introduction to the parameters and processes governing the absorption, distribution and retention of drug compounds in the body, now expanded to cover prodrugs, antitumor drugs and predictive approaches.
Synopsis: In this new edition of a bestseller, all the contents have been brought upto-date by addressing current standards and best practices in the assessment and prediction of ADMET properties. Although the previous chapter layout has been retained, substantial revisions have been made, with new topics such as pro-drugs, active metabolites and transporters covered in detail in a manner useful to the Drug Discovery scientist. The authors discuss the parameters and processes important for the absorption, distribution and retention of drug compounds in the body, plus the potential problems created by their transformation into toxic byproducts. While aimed at all those dealing professionally with the development and application of pharmaceutical substances, the readily comprehensible style makes this book equally suitable for students of pharmacy and related subjects. Uniquely comprehensive, the book relates physicochemistry and chemical structure to pharmacokinetic properties and ultimately drug efficacy and safety.
Publication: Germany
Imprint: Wiley-VCH Verlag GmbH
Returns: Returnable
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3D QSAR IN DRUG DESIGN (HB)
3D QSAR IN DRUG DESIGN (HB)
3D QSAR IN DRUG DESIGN (PB)
3D QSAR IN DRUG DESIGN (PB)
3D QSAR IN DRUG DESIGN (PB)
ANTIVIRAL DRUG STRATEGIES (HB)
ANTIVIRAL DRUG STRATEGIES, VOLUME 50
ANTIVIRAL DRUG STRATEGIES, VOLUME 50
ANTIVIRAL DRUG STRATEGIES, VOLUME 50
ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS (HB)
ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS, VOLUME 45
ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS, VOLUME 45
ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS, VOLUME 45
ATTRITION IN THE PHARMACEUTICAL INDUSTRY
ATTRITION IN THE PHARMACEUTICAL INDUSTRY
ATTRITION IN THE PHARMACEUTICAL INDUSTRY
ATTRITION IN THE PHARMACEUTICAL INDUSTRY (HB)
BIO-NMR IN DRUG RESEARCH (HB)
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54 (HB)
BIONMR IN DRUG RESEARCH, VOLUME 16
CHEMOGENOMICS IN DRUG DISCOVERY
CHEMOINFORMATICS IN DRUG DISCOVERY (HB)
CHEMOINFORMATICS IN DRUG DISCOVERY, VOLUME 23
DRUG BIOAVAILABILITY (HB)
DRUG METABOLISM PREDICTION, VOLUME 63
DRUG METABOLISM PREDICTION, VOLUME 63
DRUG METABOLISM PREDICTION, VOLUME 63
DRUG METABOLISM PREDICTION, VOLUME 63 (HB)
EVOLUTIONARY ALGORITHMS IN MOLECULAR DESIGN, VOLUME 8
FRAGMENT-BASED DRUG DISCOVERY (HB)
HIGH-THROUGHPUT SCREENING IN DRUG DISCOVERY
HIGH-THROUGHPUT SCREENING IN DRUG DISCOVERY (HB)
HIGH-THROUGHPUT SCREENING IN DRUG DISCOVERY, VOLUME 35
IN VIVO MODELS FOR DRUG DISCOVERY (HB)
LEAD GENERATION
LEAD GENERATION
LEAD GENERATION
LIGAND DESIGN FOR G PROTEIN-COUPLED RECEPTORS
LIGAND DESIGN FOR G PROTEIN-COUPLED RECEPTORS (HB)
LIGAND DESIGN FOR G PROTEIN-COUPLED RECEPTORS, VOLUME 30
METABOLISM, PHARMACOKINETICS AND TOXICITY OF FUNCTIONAL GROUPS (HB)
METABOLITE SAFETY IN DRUG DEVELOPMENT
METABOLITE SAFETY IN DRUG DEVELOPMENT
METABOLITE SAFETY IN DRUG DEVELOPMENT (HB)
MOLECULAR DESIGN (PB)
MOLECULAR DRUG PROPERTIES
MOLECULAR DRUG PROPERTIES (HB)
MOLECULAR INTERACTION FIELDS
MOLECULAR INTERACTION FIELDS (HB)
NATURAL PRODUCTS IN MEDICINAL CHEMISTRY (HB)
NATURAL PRODUCTS IN MEDICINAL CHEMISTRY, VOLUME 60
NATURAL PRODUCTS IN MEDICINAL CHEMISTRY, VOLUME 60
NATURAL PRODUCTS IN MEDICINAL CHEMISTRY, VOLUME 60
NEW TRENDS IN SYNTHETIC MEDICINAL CHEMISTRY, VOLUME 7
PAIN THERAPEUTICS
PHARMACOKINETICS AND METABOLISM IN DRUG DESIGN, VOLUME 31
PHARMACOKINETICS AND METABOLISM IN DRUG DESIGN, VOLUME 51
PHARMACOKINETICS AND METABOLISM IN DRUG DESIGN, VOLUME 51
PHARMACOKINETICS AND METABOLISM IN DRUG DESIGN, VOLUME 51
PREDICTIVE TOXICOLOGY (HB)
PRODRUGS AND TARGETED DELIVERY
PRODRUGS AND TARGETED DELIVERY
PRODRUGS AND TARGETED DELIVERY
PRODRUGS AND TARGETED DELIVERY (HB)
PROTEIN-LIGAND INTERACTIONS (HB)
PROTEIN-LIGAND INTERACTIONS, VOLUME 53
PROTEIN-LIGAND INTERACTIONS, VOLUME 53
PROTEIN-LIGAND INTERACTIONS, VOLUME 53
PROTEIN-PROTEIN INTERACTIONS IN DRUG DISCOVERY (HB)
PROTEIN-PROTEIN INTERACTIONS IN DRUG DISCOVERY, VOLUME 56
PROTEIN-PROTEIN INTERACTIONS IN DRUG DISCOVERY, VOLUME 56
PROTEIN-PROTEIN INTERACTIONS IN DRUG DISCOVERY, VOLUME 56
QSAR
REACTIVE DRUG METABOLITES (HB)
REACTIVE DRUG METABOLITES, VOLUME 55
REACTIVE DRUG METABOLITES, VOLUME 55
REACTIVE DRUG METABOLITES, VOLUME 55
SCAFFOLD HOPPING IN MEDICINAL CHEMISTRY (HB)
SCAFFOLD HOPPING IN MEDICINAL CHEMISTRY, VOLUME 58
SCAFFOLD HOPPING IN MEDICINAL CHEMISTRY, VOLUME 58
SCAFFOLD HOPPING IN MEDICINAL CHEMISTRY, VOLUME 58
THE EVOLUTION OF DRUG DISCOVERY (HB)
TRANSPORTERS AS DRUG TARGETS (HB)
VIRTUAL SCREENING
VIRTUAL SCREENING
VIRTUAL SCREENING
VIRTUAL SCREENING (HB)
VIRTUAL SCREENING FOR BIOACTIVE MOLECULES, VOLUME 10

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