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Item Details
Title: THERMODYNAMICS AND KINETICS OF DRUG BINDING, VOLUME 65
By: Gyorgy Keseru (Editor)
Format: Electronic book text

List price: £120.00


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ISBN 10: 3527673040
ISBN 13: 9783527673049
Publisher: JOHN WILEY AND SONS LTD
Pub. date: 28 July, 2015
Series: Methods and Principles in Medicinal Chemistry
Pages: 360
Synopsis: This practical reference for medicinal and pharmaceutical chemists combines the theoretical background with modern methods as well as applications from recent lead finding and optimization projects. Divided into two parts on the thermodynamics and kinetics of drug-receptor interaction, the text provides the conceptual and methodological basis for characterizing binding mechanisms for drugs and other bioactive molecules. It covers all currently used methods, from experimental approaches, such as ITC or SPR, right up to the latest computational methods. Case studies of real-life lead or drug development projects are also included so readers can apply the methods learned to their own projects. Finally, the benefits of a thorough binding mode analysis for any drug development project are summarized in an outlook chapter written by the editors.
Publication: UK
Imprint: Wiley-VCH Verlag GmbH
Returns: Non-returnable
Some other items by this author:
ADVANCED COMPUTER-ASSISTED TECHNIQUES IN DRUG DISCOVERY, VOLUME 3
ANIMAL MODELS FOR HUMAN CANCER
ANIMAL MODELS FOR HUMAN CANCER
ANIMAL MODELS FOR HUMAN CANCER
ANIMAL MODELS FOR HUMAN CANCER (HB)
ANTITARGETS
ANTITARGETS (HB)
ANTIVIRAL DRUG STRATEGIES (HB)
ANTIVIRAL DRUG STRATEGIES, VOLUME 50
ANTIVIRAL DRUG STRATEGIES, VOLUME 50
ANTIVIRAL DRUG STRATEGIES, VOLUME 50
ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS (HB)
ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS, VOLUME 45
ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS, VOLUME 45
ASPARTIC ACID PROTEASES AS THERAPEUTIC TARGETS, VOLUME 45
BIO-NMR IN DRUG RESEARCH (HB)
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54
BIOISOSTERES IN MEDICINAL CHEMISTRY, VOLUME 54 (HB)
BIONMR IN DRUG RESEARCH, VOLUME 16
CHEMOGENOMICS IN DRUG DISCOVERY
CHEMOINFORMATICS IN DRUG DISCOVERY (HB)
CHEMOINFORMATICS IN DRUG DISCOVERY, VOLUME 23
CHEMOKINE RECEPTORS AS DRUG TARGETS (HB)
CHEMOMETRIC METHODS IN MOLECULAR DESIGN, VOLUME 2
CHIRALITY IN DRUG RESEARCH, VOLUME 33
CHIRALITY IN DRUG RESEARCH, VOLUME 33 (HB)
COMBINATORIAL CHEMISTRY
COMBINATORIAL CHEMISTRY
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DRUG BIOAVAILABILITY
DRUG BIOAVAILABILITY (HB)
DRUG METABOLISM PREDICTION, VOLUME 63
DRUG METABOLISM PREDICTION, VOLUME 63
DRUG METABOLISM PREDICTION, VOLUME 63
DRUG METABOLISM PREDICTION, VOLUME 63 (HB)
DRUG SELECTIVITY
DRUG-MEMBRANE INTERACTIONS
EPIGENETIC TARGETS IN DRUG DISCOVERY
EPIGENETIC TARGETS IN DRUG DISCOVERY (HB)
EPIGENETIC TARGETS IN DRUG DISCOVERY, VOLUME 42 (HB)
EVOLUTIONARY ALGORITHMS IN MOLECULAR DESIGN, VOLUME 8
FRAGMENT-BASED APPROACHES IN DRUG DISCOVERY
FRAGMENT-BASED APPROACHES IN DRUG DISCOVERY, VOLUME 34
FRAGMENT-BASED APPROACHES IN DRUG DISCOVERY, VOLUME 34 (HB)
FRAGMENT-BASED DRUG DISCOVERY
FRAGMENT-BASED DRUG DISCOVERY
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G PROTEIN-COUPLED RECEPTORS AS DRUG TARGETS
G PROTEIN-COUPLED RECEPTORS AS DRUG TARGETS (HB)
HANDBOOK OF MOLECULAR DESCRIPTORS, VOLUME 11
HIGH-THROUGHPUT SCREENING IN DRUG DISCOVERY
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HIT AND LEAD PROFILING (HB)
HOW TO PASS NATIONAL 5 ENGLISH (PB)
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IN VIVO MODELS FOR DRUG DISCOVERY (HB)
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LEAD GENERATION
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LIGAND DESIGN FOR G PROTEIN-COUPLED RECEPTORS
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MASS SPECTROMETRY IN MEDICINAL CHEMISTRY
MASS SPECTROMETRY IN MEDICINAL CHEMISTRY
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MEDICINAL CHEMISTRY APPROACHES TO PERSONALIZED MEDICINE (HB)
MEDICINAL CHEMISTRY APPROACHES TO PERSONALIZED MEDICINE, VOLUME 59
MEDICINAL CHEMISTRY APPROACHES TO PERSONALIZED MEDICINE, VOLUME 59
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MICROWAVES IN ORGANIC AND MEDICINAL CHEMISTRY
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MOLECULAR DESCRIPTORS FOR CHEMOINFORMATICS (HB)
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MOLECULAR DRUG PROPERTIES
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MOLECULAR INTERACTION FIELDS
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MOLECULAR MODELING
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NATURAL PRODUCTS IN MEDICINAL CHEMISTRY, VOLUME 60
NATURAL PRODUCTS IN MEDICINAL CHEMISTRY, VOLUME 60
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PRACTICE PAPERS INTERMEDIATE 2 ENGLISH (PB)
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PROTEIN-LIGAND INTERACTIONS
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PROTEIN-LIGAND INTERACTIONS, VOLUME 53
PROTEIN-PROTEIN INTERACTIONS IN DRUG DISCOVERY (HB)
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QSAR
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